至今,GenScript的服务及产品已被Cell, Nature, Science, PNAS等1300多家生物医药类杂志引用近万次,处于行业领先水平。NIH、哈佛、耶鲁、斯坦福、普林斯顿、杜克大学等约400家全球著名机构使用GenScript的基因合成、多肽服务、抗体服务和蛋白服务等成功地发表科研成果,再次证明GenScript 有能力帮助业内科学家Make research easy.

Discovery of Novel Potent Muscarinic M3 Receptor Antagonists with Proper Plasma Stability by Structural Recombination of Marketed M3 Antagonists

ChemMedChem. 2017; 
Zuojuan Xiang+ , Jun Liu+ , Hongbin Sun,* and Xiaoan Wen*[a]
Products/Services Used Details Operation
Cellular Analysis All binding assays were performed in 96-well plates (UniFilter 96 GF/C, PerkinElmer) with membrane preparation expressing human M3 receptors (transfected CHO-K1 cells, GenScript USA Inc.). Get A Quote

摘要

关键词

ammonium salts · antagonists · nitrogen heterocycles · stability · structure–activity relationships